您好,欢迎访问三七文档
当前位置:首页 > 行业资料 > 其它行业文档 > 从基因到天然产物生物合成
There-emergenceofnaturalproductsfordrugdiscoveryinthegenomicsera药物基因组学教研室解鸿波NaturalproductsanddrugdiscoveryNaturalproductsandgenomicsFuturedirectionsandoutlookSourcesofNaturalproducts1234Whatarenaturalproducts?1.SourcesofNaturalproductsWhatarenaturalproducts?1.SourcesofNaturalproductsArtemisinin2.NaturalproductsanddrugdiscoveryMorphineQuininePaclitaxel6%27%25%5%37%AllsmallmoleculenewchemicalentitiesCommerciallyavailablechemicalspace22x106compoundsNaturalproductuniverse16x104compoundsNatural-productdatabasesDatabaseNumberofentriesAdditionalinformationSuperNaturalII355,0002DstructureswithvendorinformationUniversalNaturalProductDatabase197,2013DstructuresassembledfromotherdatabasesChineseNaturalProductDatabase53,000HasbeenusedinvirtualscreeniSMART20,000FromtraditionalChinesemedicinesAfroDb1,000FromAfricanmedicinalplantsInteractionsbetweendrugandtarget3.NaturalproductsandgenomicsInsightsintotheBiosynthesisInsightsintotheBiosynthesisGeneclusterBioinformaticstoolsantiSMASH3.0DiscovernewdrugleadsDiscovernewdrugleadsPromoterreplacementsandgenedeletions4.Futuredirectionsandoutlook“Therewasanintrinsicbeliefinthevalueofthemoleculeswe'reseeking.”–GregoryVerdine
本文标题:从基因到天然产物生物合成
链接地址:https://www.777doc.com/doc-5301586 .html